Bioactive molecules
Cell Cycle/DNA Damage
Antifolate
APC
ATM/ATR
Aurora Kinase
Casein Kinase
CDK
CRISPR/Cas9
Deubiquitinase
DNA-PK
Checkpoint Kinase (Chk)
DNA Alkylator/Crosslinker
DNA/RNA Synthesis
Eukaryotic Initiation Factor (eIF)
G-quadruplex
Haspin Kinase
HDAC
HSP
IRE1
Kinesin
LIM Kinase (LIMK)
Microtubule/Tubulin
Mps1
Nucleoside Antimetabolite/Analog
p97
PAK
PARP
PERK
Polo-like Kinase (PLK)
PPAR
RAD51
ROCK
Sirtuin
SRPK
Telomerase
TOPK
Topoisomerase
Wee1
GPCR/G Protein
5-HT Receptor
Adenosine Receptor
Adenylate Cyclase
Adiponectin Receptor
Adrenergic Receptor
Angiotensin Receptor
Bombesin Receptor
Bradykinin Receptor
Cannabinoid Receptor
CaSR
CCR
CGRP Receptor
Cholecystokinin Receptor
CRFR
CXCR
Dopamine Receptor
EBI2/GPR183
Endothelin Receptor
GHSR
Glucagon Receptor
Glucocorticoid Receptor
GNRH Receptor
GPCR19
GPR109A
GPR119
GPR120
GPR139
GPR40
GPR55
GPR84
Guanylate Cyclase
Histamine Receptor
Imidazoline Receptor
Leukotriene Receptor
LPL Receptor
mAChR
MCHR1 (GPR24)
Melanocortin Receptor
Melatonin Receptor
mGluR
Motilin Receptor
Neurokinin Receptor
Neuropeptide Y Receptor
Neurotensin Receptor
Opioid Receptor
Orexin Receptor (OX Receptor)
Oxytocin Receptor
P2Y Receptor
Prostaglandin Receptor
Protease-Activated Receptor (PAR)
Ras
RGS Protein
Sigma Receptor
Somatostatin Receptor
TSH Receptor
Urotensin Receptor
Vasopressin Receptor
Membrane Transporter/Ion Channel
ATP Synthase
BCRP
Calcium Channel
CFTR
Chloride Channel
CRAC Channel
CRM1
EAAT2
GABA Receptor
GlyT
HCN Channel
iGluR
Monoamine Transporter
Monocarboxylate Transporter
Na+/Ca2+ Exchanger
Na+/HCO3- Cotransporter
Na+/K+ ATPase
nAChR
NKCC
P-glycoprotein
P2X Receptor
Potassium Channel
Proton Pump
SGLT
Sodium Channel
TRP Channel
URAT1
Metabolic Enzyme/Protease
15-PGDH
5 alpha Reductase
5-Lipoxygenase
Acetyl-CoA Carboxylase
Acyltransferase
Adenosine Deaminase
Adenosine Kinase
Aldehyde Dehydrogenase (ALDH)
Aldose Reductase
Aminoacyl-tRNA Synthetase
Aminopeptidase
Angiotensin-converting Enzyme (ACE)
Arginase
ATGL
ATP Citrate Lyase
Carbonic Anhydrase
Carboxypeptidase
Cathepsin
COMT
Drug Metabolite
Elastase
Endogenous Metabolite
Enolase
FAAH
FABP
Factor Xa
Farnesyl Transferase
Fatty Acid Synthase (FAS)
FXR
Glucokinase
Glutathione Peroxidase
GSNOR
Gutathione S-transferase
HCV Protease
Hexokinase
HIV Integrase
HIV Protease
HIF/HIF Prolyl-Hydroxylase
HMG-CoA Reductase (HMGCR)
HSP
Indoleamine 2,3-Dioxygenase (IDO)
Isocitrate Dehydrogenase (IDH)
Lactate Dehydrogenase
LXR
MAGL
MALT1
Mineralocorticoid Receptor
Mitochondrial Metabolism
MMP
Nampt
NEDD8-activating Enzyme
Neprilysin
PAI-1
PDHK
PGC-1α
Phosphatase
Phosphodiesterase (PDE)
Phospholipase
Procollagen C Proteinase
Proteasome
Pyruvate Kinase
RAR/RXR
Renin
ROR
Ser/Thr Protease
SGK
Stearoyl-CoA Desaturase (SCD)
Thrombin
Tryptophan Hydroxylase
Tyrosinase
Xanthine Oxidase
Neuronal Signaling
CGRP Receptor
COMT
5-HT Receptor
AChE
Adenosine Kinase
Amyloid-β
Beta-secretase
CaMK
Dopamine Receptor
Dopamine Transporter
FAAH
GABA Receptor
GlyT
iGluR
Imidazoline Receptor
mAChR
Melanocortin Receptor
Melatonin Receptor
Monoamine Oxidase
nAChR
Neurokinin Receptor
Opioid Receptor
Serotonin Transporter
γ-secretase
API
Intermediates
Others
| Catalog No. | Cas No. | Chemical name |
| ATK-A00182 | 130089-98-4 | |
| ATK-A00488 | 91396-88-2 | |
| ATK-A00192 | 80306-38-3 | |
| ATK-A00220 | 1260075-17-9 | |
| ATK-A00280 | 101155-02-6 | |
| ATK-A00094 | 292135-78-5 | |
| ATK-A00103 | 445295-04-5 | |
| ATK-A00476 | 947620-48-6 | |
| ATK-A00127 | 1238697-26-1 | |
| ATK-A00340 | 1144035-53-9 |
